Compile Data Set for Download or QSAR
maximum 50k data
Found 10 of affinity data for UniProtKB/TrEMBL: Q2FXH2
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286770(CHEMBL4171058)
Affinity DataIC50:  640nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286767(CHEMBL4172643)
Affinity DataIC50:  650nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286774(CHEMBL4163140)
Affinity DataIC50:  920nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286768(CHEMBL4171458)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286765(CHEMBL4159778)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286771(CHEMBL4167692)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286775(CHEMBL4174152)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286766(CHEMBL4163450)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286772(CHEMBL4160841)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286769(CHEMBL4161986)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed